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5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol
Ingredients/Compound/5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol.

Strength pending.The research strength is not set yet.

A plant stilbene in the resveratrol family. Its phenol groups hand a hydrogen atom to radical species, which is the chemistry behind how this class behaves as an antioxidant.

HECompound
5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diolIngredientMD
Category
Compound

What 5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol is, and what it does.

Does it work
Suits a formulator who wants the stilbene chemistry named precisely. Only 2 records carry this exact name, so read it as the class rather than a separate story.
How much to take
No dose figure is on record for this compound. Stilbenes dissolve poorly, so a daily amount taken with fat or in a phospholipid form is what actually gets absorbed.
Time to feel it
Nobody has measured a human time course under this name. Stilbenes peak in blood within a couple of hours, mostly as conjugates rather than the free molecule.
The first dose
Day one is an absorption story. What reaches your blood in the first hours is largely glucuronide and sulfate conjugate, and no sensation is described.
With regular use
Weeks of daily use have not been studied under this exact name. Where change would show is in oxidative stress markers on a lab panel rather than in a given day.
How well tolerated
No human safety dataset sits under this name. Stilbenes as a class are well tolerated at supplement amounts, and anyone on blood-thinning medication should ask a doctor.
How it feels
Nobody has described a subjective effect. Where this class registers is a laboratory antioxidant marker rather than anything you would notice.
The overlooked benefit
Ultraviolet light flips the stable trans form to cis, so a clear bottle on a sunny shelf changes what is inside. Opaque packaging is doing real work here.

The proof, claim by claim.

These words describe the research, not the molecule's worth. Research strength is how much work stands behind one claim, and it is never a product score.

  • Radical scavenging by phenolic stilbenesIn vitro study
  • First-pass conjugation limiting stilbene bioavailabilityNarrative review
  • Stilbene production by plants as a phytoalexin responseNarrative review
  • Light-driven isomerisation of the trans formIn vitro study
PubMedCochraneClinicalTrials.govNIH ODSSUPP.AILabs test. IngredientMD verifies.PubMedCochraneClinicalTrials.govNIH ODSSUPP.AILabs test. IngredientMD verifies.
Pairs well with7 on file

Why these belong in the same formula. Each row says what the basis is, from settled biochemistry through to a trial that measured the pair.

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol + QuercetinShared phase II conjugation enzymes, established competition

Both this stilbene and quercetin are substrates for the same UDP-glucuronosyltransferase and sulfotransferase isoforms in the gut wall and liver. Co-dosing loads those enzymes and can raise circulating free concentrations of either compound. That is a pharmacokinetic interaction rather than a demonstrated benefit, and it cuts both ways.

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol + ResveratrolStructural isomerism and shared metabolic handling

This compound is a trihydroxystilbene closely related to resveratrol, differing in the position of the phenolic hydroxyls. It goes through the same rapid glucuronidation and sulfation on first pass, which is why systemic exposure to any of these stilbenes is low relative to the dose taken. Combining them does not solve that problem, it shares it.

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol + Vitamin CEstablished phenoxyl radical reduction chemistry

When a phenolic compound quenches a radical it becomes a phenoxyl radical itself. Ascorbate reduces that species back to the parent phenol, which is standard antioxidant network chemistry and applies to stilbenes as a class. It describes behaviour in solution, not a measured outcome in a person.

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol + Sunflower LecithinPhospholipid dispersion of poorly water-soluble polyphenols

Stilbenes are lipophilic and dissolve poorly in gut fluid, which limits how much can be presented for absorption. Phospholipid complexes and lecithin dispersions raise apparent solubility and are a standard formulation answer for this class. The gain is in dissolution, and dissolution is only one of the barriers.

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol + Black Pepper Extract (BioPerine)Piperine inhibition of glucuronidation, established for polyphenols

Piperine inhibits intestinal UGT activity, and glucuronidation is the main reason stilbene blood levels stay low after an oral dose. Pairing the two raises systemic exposure of the parent compound. The same inhibition applies to co-administered drugs, which is why the pairing is not a free lunch.

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol + MCT OilLipid vehicle effect on lipophilic phenolics

Taking a lipophilic polyphenol with a fat source stimulates bile release and micelle formation, which puts more of the compound into an absorbable state. Fasted dosing of a dry stilbene powder is the worst case for uptake. This is general lipophilic-nutrient handling applied to the class.

5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol + ProbioticsGut microbial conversion of stilbene glycosides

Stilbenes often arrive in plant material as glycosides, and gut bacterial glycosidases cleave the sugar to release the free aglycone that can cross the enterocyte. Which bacteria are present therefore shapes how much free compound is generated. Individual conversion capacity varies widely and is not routinely measured.

Who should be cautious

Nothing specific on file for 5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol. Match the label to the daily amount above, and tell your doctor what you take.

Not medical advice. Show the label to your pharmacist.

What 5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol actually does.

Established

This compound is a stilbene with three hydroxyl groups spread across two connected rings.

Established

The central double bond can exist in two shapes. The more stable shape can flip to the other under ultraviolet light, which is why stilbene materials are kept away from light.

Established

Phenolic hydroxyl groups on this stilbene donate a hydrogen atom to neutralise free radicals, forming a stable radical themselves. This is the chemical basis for stilbene antioxidant activity seen in the lab.

Established

Stilbenes get heavily modified in the gut wall and liver before entering circulation, so most of what's in blood after an oral dose is a modified form rather than the original compound.

More than one route, 6 steps on record

Where 5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol comes from.

It is a small plant-type molecule in the same family as resveratrol. It can be made in a factory or pulled out of plants, and either way it has to be kept in the dark because light changes its shape.

The same molecule is reached more than one way. Which route a given product used is a manufacturing choice, and the finished compound is the same either way.

Starts as
Plant material or petrochemical starting blocks

The botanical route uses stilbene-accumulating plant tissue such as vine, root or bark. The synthetic route starts from substituted benzaldehydes and phosphonium or phosphonate reagents.

Converted by
Wittig or Heck coupling for the synthetic route

The stilbene double bond is formed by a Wittig-type olefination or a palladium-catalysed Heck coupling between an aryl halide and a styrene, followed by removal of protecting groups from the phenols.

Extracted by
Solvent extraction for the botanical route

Ethanol or ethyl acetate pulls the stilbene fraction from milled plant material. Yields are low because plants make these compounds only in small amounts and mostly under stress.

Purified by
Recrystallisation or chromatography

Recrystallisation removes reaction by-products and non-target polyphenols. Column chromatography is used where a single isomer at high purity is required.

Standardised to
HPLC assay of the trans isomer

Purity and isomer ratio are set by high performance liquid chromatography with ultraviolet detection, since the cis and trans forms separate cleanly and absorb differently.

Ends up as
Light-protected powder

Packed in amber or opaque containers under low humidity, because ultraviolet exposure drives trans to cis conversion and moisture accelerates degradation.

Getting 5-[2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol from food.

The whole-food sources on file. A supplement closes the gap, it does not replace dinner.

Red grape skinsRed winePeanutsBlueberries

A gram-for-gram figure (how much of each you would eat to match a dose) will appear here once it is sourced and reviewed. This page will not print a number it cannot cite.

The forms it comes in.

Stilbene glucosideA sugar unit attached at a phenolic hydroxyl, which raises water solubility considerablyFits Aqueous formats and plant extracts where the glycoside is the native formTrade-off Requires gut bacterial or brush-border glycosidase cleavage before the active aglycone is released, and that capacity varies between people
Phospholipid-complexed stilbeneThe phenol is associated with phosphatidylcholine, creating an amphipathic complexFits Formulas where dissolution is the limiting step and a higher plasma level is the design goalTrade-off Bulkier per unit of active, more expensive per gram, and does nothing about phase II conjugationActive and formulation aid
Stilbene in beta-cyclodextrinThe lipophilic core sits inside the cyclodextrin cavity while the outer surface stays hydrophilicFits Beverages and rapidly dissolving powders, and it also shields the compound from light-driven isomerisationTrade-off The carrier adds substantial mass, so declared complex weight is far higher than active weightActive and formulation aid
Stilbene-standardised botanical extractA mixed polyphenol matrix with the target stilbene assayed to a stated percentageFits Whole-matrix formulations where the accompanying polyphenols are considered part of the materialTrade-off Other stilbenes and flavonoids ride along uncounted, which makes the actual dose of any one molecule less certain

FDA Disclaimer: These statements have not been evaluated by the Food and Drug Administration. This information is for educational purposes only and is not intended to diagnose, treat, cure, or prevent any disease. Consult your healthcare provider before starting any supplement regimen.